Co-reporter: Tingting Mo, Xueling Mi, Erin E. Milner, Geoffrey S. Dow, Peter Wipf
pp: 5137-5140
Publication Date(Web):29 September 2010
DOI: 10.1016/j.tetlet.2010.07.113
The 8-SF5 analog of mefloquine was synthesized in nine steps from commercially available starting materials and in five steps from a novel ortho-SF5–substituted aniline intermediate.